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Synthesis of a Library of 1,5,2-Dithiazepine 1,1-Dioxides. Part 1: A One-Pot Sulfonylation/Thia-Michael Protocol

dc.contributor.authorZang, Qin
dc.contributor.authorZhou, Aihua
dc.contributor.authorJaved, Salim
dc.contributor.authorMaity, Pradip K.
dc.contributor.authorKnudtson, Christopher Anton
dc.contributor.authorBi, Danse
dc.contributor.authorHastings, Jared J.
dc.contributor.authorBasha, Fatima Z.
dc.contributor.authorHanson, Paul R.
dc.date.accessioned2017-06-13T15:35:38Z
dc.date.available2017-06-13T15:35:38Z
dc.date.issued2012-12-31
dc.identifier.citationZang, Q., Zhou, A., Javed, S., Maity, P. K., Knudtson, C. A., Bi, D., … Hanson, P. R. (2012). Synthesis of a Library of 1,5,2-Dithiazepine 1,1-Dioxides. Part 1: A One-Pot Sulfonylation/Thia-Michael Protocol. Heterocycles, 86(2), 10.3987/COM–12–S(N)121. http://doi.org/10.3987/COM-12-S(N)121en_US
dc.identifier.urihttp://hdl.handle.net/1808/24480
dc.description.abstractA novel one-pot sulfonylation/intramolecular thia-Michael protocol is reported for the synthesis of 1,5,2-dithiazepine 1,1-dioxides. Sulfonylation between cysteine ethyl ester/cysteamine and 2-chloroethanesulfonyl chloride, followed by in situ intramolecular thia-Michael addition, was achieved and afforded the titled 1,5,2-dithiazepine-1,1-dioxide scaffolds. Diversification was demonstrated for future library synthesis.en_US
dc.publisherElsevieren_US
dc.rightsThis is an open access article under the terms of the Creative Commons Attribution-NonCommercial-NoDerivs License 4.0 (CC BY-NC-ND 4.0), which permits use and distribution in any medium, provided the original work is properly cited, the use is non-commercial and no modifications or adaptations are made.en_US
dc.rights.urihttp://creativecommons.org/licenses/by-nc-nd/4.0/en_US
dc.titleSynthesis of a Library of 1,5,2-Dithiazepine 1,1-Dioxides. Part 1: A One-Pot Sulfonylation/Thia-Michael Protocolen_US
dc.typeArticleen_US
kusw.kuauthorZang, Qin
kusw.kuauthorZhou, Aihua
kusw.kuauthorJaved, Salim
kusw.kuauthorMaity, Pradip K.
kusw.kuauthorKnudtson, Chris A.
kusw.kuauthorBi, Danse
kusw.kuauthorHastings, Jared J.
kusw.kuauthorHanson, Paul R.
kusw.kudepartmentChemistryen_US
dc.identifier.doi10.3987/COM-12-S(N)121.en_US
kusw.oaversionScholarly/refereed, author accepted manuscripten_US
kusw.oapolicyThis item meets KU Open Access policy criteria.en_US
dc.identifier.pmidPMC3873773en_US
dc.rights.accessrightsopenAccess


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This is an open access article under the terms of the Creative Commons Attribution-NonCommercial-NoDerivs License 4.0 (CC BY-NC-ND 4.0), which permits use and distribution in any medium, provided the original work is properly cited, the use is non-commercial and no modifications or adaptations are made.
Except where otherwise noted, this item's license is described as: This is an open access article under the terms of the Creative Commons Attribution-NonCommercial-NoDerivs License 4.0 (CC BY-NC-ND 4.0), which permits use and distribution in any medium, provided the original work is properly cited, the use is non-commercial and no modifications or adaptations are made.