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    Design, Synthesis and Evaluation of Peptide-Based Affinity Labels for Mu Opioid Receptors (1)
    DESIGN, SYNTHESIS AND METABOLISM OF ARODYN ANALOGS (1)
    Design, Synthesis, and Evaluation of Site-Specific Hsp90 Inhibitors (1)
    Development of a Parallel Strategy for the Synthesis of a Library of 2-(3-Formyl-5-arylfuran-2-yl)ethylcarbamates from Dihydropyridinones (1)
    Development of libraries inspired by sparteine (1)
    Development of Three Reaction Methodologies En Route to Nitrogen Containing Heterocycles: a Diels-Alder/Schmidt, a DIels-Alder/Acylation and a Catalytic Intramolecular Schmidt (1)
    Discovery of Novel Inhibitors of Cellular Efflux by High-Content Screening with a Fluorescent Mimic of Taxol (1)
    Diverse Applications of Flow Technology in Discovery Chemistry (1)
    Exploration of Salvinorin A for the Development of Pain and Addiction Therapies (1)
    Exploration of the Mechanisms of Adjuvanticity for Toll-like Receptor Agonists (1)
    Exploration of Toll-like Receptor 7 and 8 Agonists as Potential Vaccine Adjuvants (1)
    Human Cytochrome P450 2E1: Functional Comparison to Cytochrome 2A13 and 2A6 (1)
    I. Catalysis of Intra- and Intermolecular Schmidt Reactions. II. Copper-Catalyzed Oxaziridine-Mediated C-H Bond Oxidation. III. Synthesis and Cytotoxic Evaluation of Withalongolide A Analogues. (1)
    I. Development of Bisamides as Kappa Opioid Receptor Agonists. II. Potency Enhancement of Sulfonamide-based Kappa Opioid Receptor Antagonists. III. Asymmetric Acyl Transfer Reactions Catalyzed by a Cyclic Peptide. (1)
    I. Selective Probes for Cytochrome P450 17A1 Suggest a Design Strategy Toward Improved Breast and Prostate Cancer Agents II. Spatiotemporal Control of Reactivity via Visible Light-Mediated C-H Activation Creates Patterned Carbohydrate Surfaces III. Toward Catalytic Intramolecular Schmidt Reactions (1)
    Improving the Yeast Three-Hybrid System for High-Throughput Target Discovery (1)
    Inhibition of Heat Shock Protein 90 Machinery for the Treatment of Cancer: Progress in the Development of Alternative Strategies (1)
    Investigation of Natural Product Scaffolds for the Development of Opioid Receptor Ligands (1)
    Investigation of the Hsp90 C-terminal Binding Site, Novel Inhibitors and Isoform-Dependent Client Proteins (1)
    Investigation of the Phenyl Ring of Imidazoquinolines (1)
    Investigations Of Salvinorin A: Synthetic Isolation, Quantification, And In Vivo Characteristics (1)
    Iron-catalyzed decarboxylative cross coupling reactions and palladium-catalyzed sp2-sp3 coupling of coumarins. (1)
    Isatin Derivatives as Inhibitors of Microtubule Assembly (1)
    Modulators of Toll-like Receptors -7 and -8 (1)
    Modulators of Toll-like Receptors-4 and -2 (1)
    Natural Product Inhibitors of Hsp90: Potential Leads for Drug Discovery (1)
    Novel Intramolecular Nucleophilic Addition Reactions: Formation of Unusual N-O-Heterocyclic Enones (1)
    Nucleophilic Additions to 3-Azido-hexanal (1)
    Part I. Approaches Toward the Total Synthesis of Tyloindicine F; Part II. Palladium-Catalyzed C−H Functionalization of β-enaminones (1)
    Phase-Trafficking Methods in Natural Products, Modulators of Organic Anion Transporting Polypeptides from Rollinia emarginata, and Pregnane and Cardiac Glycosides from Asclepias spp. (1)
    Phenanthropiperidine Alkaloids: Methodology Development, Synthesis and Biological Evaluation (1)
    Probing the Antibiotic Target MurA from S. aureus and B. subtilis (1)
    Stereodivergent Synthesis of Enantioenriched Five- and Six-Membered Cyclic-1,3-diols and Applications Toward Library Synthesis (1)
    Strategies for the Fluorine-Retentive Functionalization of Gem-Difluoroalkenes (1)
    Structural and Functional Evaluation of Steroidogenic Cytochrome P450 Enzymes (1)
    Structure-Based Design of Grp94-Selective Inhibitors (1)
    Studies and Synthetic Methodology: 1. Cycloaddition of Allylic Azides and Alkynes, 2. Hexafluoro-2-propanol-promoted Friedel–Crafts Acylation Reactions (1)
    STUDIES OF INTERACTIONS OF SMALL MOLECULES WITH MEMBRANES AND PROTEINS (1)
    Studies of novel targeted drug delivery systems and molecular probes of cancer biology (1)
    Studies on Oximidine II - Total Synthesis by an Unprecedented Reductive Coupling (1)
    Synthesis and biological evaluation of dynorphin analogs and, Caco-2 permeability of opioid macrocyclic tetrapeptides (1)
    Synthesis and Evaluation of Fluorescent Tools for Studies of Cancer Biology (1)
    Synthesis and evaluation of modified oximidine analogues as anticancer agents and of terephthalaldehyde-bis-guanylhydrazones as endotoxin sequestering agents (1)
    Synthesis and Evaluation of Novel Iminosugars as Potential Male Contraceptive Agents; and the Chemistry of 2,3-Dihydropyridin-4-(1H)-ones and Related Enaminones in Multicomponent Reactions (1)
    SYNTHESIS AND PHENOTYPIC DISCOVERY OF MOLECULAR PROBES OF BIOLOGICAL SYSTEMS (1)
    Synthesis and Reactivity of Medium-Bridged Twisted Lactams (1)
    Synthetic and computational efforts toward the understanding and development of novobiocin-derived inhibitors of Hsp90 (1)
    Synthetic delivery systems that control release of anticancer agents from early endosomes (1)
    Synthetic Molecular Probes of Endocytosis, Escape from Endosomes, and Protein-Protein Interactions (1)
    Synthetic Strategies for the Lepadiformines and Cylindricine C via Tandem Schmidt Reactions (1)
    Synthetic Strategies to Access Biologically Important Fluorinated Motifs: Fluoroalkenes and Difluoroketones (1)
    The Application of X-ray Crystallography towards the Design of Novel Inhibitors of MurA and CDK2 (1)
    The Design, Synthesis and Evaluation of Peptide Ligands to Study Opioid Receptors (1)
    The Development of Organelle-localized Hsp90 Isoform-selective Inhibitors (1)
    The Development of Small Molecules that Modulate Molecular Chaperones Hsp90 and Hsp70 (1)
    The human cytochrome P450 2A family: Comparisons and identification of amino acids essential for substrate recognition (1)
    The Pursuit of Unshocking Hsp90 Inhibitors: Development of Gedunin and Cruentaren A as Chemical Leads (1)
    The Synthesis and Pharmacological Evaluation of Salvinorin A Analogues as Opioid Receptor Probes (1)
    Unfolding the Hsp90 Foldasome: Structure-Activity Relationship Studies on EGCG and Development of Isoform-Selective Inhibitors (1)
    Vinylogous Esters and Amides: Useful Synthons for Diversity-Oriented and Natural Product Synthesis (1)